Elsevier

Tetrahedron Letters

Volume 53, Issue 9, 29 February 2012, Pages 1051-1055
Tetrahedron Letters

Synthesis and cross-coupling reactions of imidomethyltrifluoroborates with aryl chlorides

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Abstract

Potassium imidomethyltrifluoroborate salts were efficiently synthesized. Potassium phthalimidomethyltrifluoroborate was successfully used in Suzuki–Miyaura-like cross-coupling reactions with a variety of aryl chlorides.

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Acknowledgments

This research was supported by a National Priorities Research Program (NPRP) grant from the Qatar National Research Fund (Grant No. 08-035-1-008). G.A.M. thanks the National Institute of General Medical Sciences for support.

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